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Updated: Jan 10, 2026

Quantitative Structure-Activity Relationship, Activity Prediction, and Molecular Dynamics of Non-nucleotide Reverse Transcriptase Inhibitors
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Published on: May 9, 2025

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多含化合物作为多位sEH/FAAH抑制剂:结构-活性关系和药理学研究

Amanda Tsang1, Cassandra Yuan1, Manuel Berumen1

  • 1Department of Chemistry & Biochemistry, California State University, Fullerton, 800 N. State College, Fullerton, CA 92834, United States.

Bioorganic & medicinal chemistry
|November 25, 2025
PubMed
概括

针对可溶性环氧化酶 (sEH) 和脂肪酸胺酶 (FAAH) 的新型双抑制剂提供非阿片类药物疼痛缓解. 这种新型的昆西尼尔类比4m显示出高强度,但可能会导致行为影响.

关键词:
酶抑制可以抑制酶.高的药物是高的药物.微小体肝脏测定方法微波辅助合成技术的使用多目标定向的带多目标定向的带.结构与活动的关系.轮子运行,轮子运行.

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