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Updated: Jan 9, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
07:16

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Published on: August 16, 2018

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与GABA效应剂相比,新型三胺-三酸的活体中神经变效应与GABA效应剂相比

Anatoly Demchenko1,2,3, Artur Martynov4, Yevhenii Novodvorskyi5

  • 1Department of Chemistry, Pontifical Catholic University of Rio de Janeiro (PUC-Rio), 225-Marquês de São Vicente St., Rio de Janeiro 22451-900, Rio de Janeiro Brazil.

ACS chemical neuroscience
|December 4, 2025
PubMed
概括

新的三胺-氨酸化合物显示出有前途的抗焦虑作用. 化合物11g在动物模型中显示出强大的焦虑减轻作用,为神经性障碍提供了潜在的新疗法.

关键词:
在13C NMR中.一个小时的NMR.自动码头 维纳码头 在 silico 码头在活体中使用抗焦虑药物.开放的实地研究研究.有机合成有机合成三胺-三氨酸-三氨酸.

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