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Updated: Jan 9, 2026

Measuring G-protein-coupled Receptor Signaling via Radio-labeled GTP Binding
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Measuring G-protein-coupled Receptor Signaling via Radio-labeled GTP Binding

Published on: June 9, 2017

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与选择性激动剂复合的G蛋白结合受体HCAR3的结构揭示了连接体识别和选择性的基础

Fang Ye1,2, Zhiyi Zhang2,3, Binghao Zhang2

  • 1Guangxi Key Laboratory of Special Biomedicine, School of Medicine, Guangxi University, Nanning, China.

PLoS biology
|December 8, 2025
PubMed
概括

碳酸受体3 (HCAR3) 的结构洞察力揭示了特定的结合机制,使其与HCAR2区别开来. 这项研究有助于开发针对HCAR3的药物,以避免HCAR2的副作用.

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