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Updated: Jan 8, 2026

Quantitative Structure-Activity Relationship, Activity Prediction, and Molecular Dynamics of Non-nucleotide Reverse Transcriptase Inhibitors
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双甲衍生物作为11β-氧类固醇脱酶的强有力的抑制剂2:结构-活性研究

Xiya Ren1, Lei Shi2, Xinyue Chen3

  • 1Department of Obstetrics and Gynecology, the Second Affiliated Hospital and Yuying Children's Hospital of Wenzhou Medical University, Wenzhou, Zhejiang 325027, China.

The Journal of steroid biochemistry and molecular biology
|December 19, 2025
PubMed
概括

双甲衍生物 (BPADs) 是一种新的11β-基类固醇脱酶2型 (11β-HSD2) 的抑制剂. 4-基甲 (BPH) 是最强效的,对内分泌干扰有影响,特别是在怀孕期间.

关键词:
11β-HSD2 的抑制.双甲基衍生物 双甲基衍生物内分泌干扰物 干扰内分泌干扰物分子对接是分子对接.结构与活动关系 (SAR)表面等离子体共振是什么?

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