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嵌合体效率在TRPA1的面向膜的部位形成了连接物接入和结合

Charles Mariasoosai1, Ayobami Diyaolu1, Peter Obi1

  • 1College of Pharmacy and Pharmaceutical Sciences, Washington State University, Spokane, Washington 99202, United States.

Journal of medicinal chemistry
|December 23, 2025
PubMed
概括

研究人员探索了TRPA1抗剂如何与细胞膜相互作用. 一个新的指标,黑效率 (CE),通过评估连接体适应性来访问膜结合部位来预测药物的效力.

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