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Updated: Jan 13, 2026

Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines
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Published on: June 23, 2019

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设计,合成和功能化的1,2,4,5-四替代-胺的抗炎活性

Rayees Ahmad Naikoo1, Diljeet Kumar2,3, Nusrit Iqbal Andrabi2,3

  • 1Department of Chemical Sciences, I.K. Gujral Punjab Technical University, Kapurthala, India.

Chemistry & biodiversity
|January 8, 2026
PubMed
概括

两个新型的胺衍生物,3d和3f通过减少炎症介质和巨细胞中的蛋白质表达,显示出强大的抗炎作用. 这些化合物代表了开发新抗炎药物的有希望的线索.

关键词:
氨基金胺氨基.它具有抗炎潜在的抗炎作用.阿扎-迈克尔的补充.α,β-不和的烯酸.这是β-氨基碳烯化合物.

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