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Updated: Jan 18, 2026

Synthesis of a Borylated Ibuprofen Derivative Through Suzuki Cross-Coupling and Alkene Boracarboxylation Reactions
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Published on: November 30, 2022

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合成和奇拉分离的布洛芬衍生品增加抗炎活性

Mohd Mustaqeem1, Ann Gogolashvili2, Lali Chankvetadze3

  • 1Department of Chemistry, Jamia Millia Islamia, New Delhi, India.

Chirality
|January 16, 2026
PubMed
概括

合成了15种新型的布洛芬衍生物,并成功将其分离成反体. 这些衍生品对COX-II具有增强的结合亲和力,这表明它们的疗效和未来药物的潜力有所提高.

关键词:
通过建模生物疗效来确定生物疗效.乙聚合物的分辨率.伊布洛芬衍生品 伊布洛芬衍生品奇拉分离的机制.合成和表征的方法.

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