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Updated: Jan 24, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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小分子激动剂和对抗剂的实施,以阐明淋巴激素受体结构,功能和生理学

James A Dias1, Claire L Newton2, Alfredo Ulloa-Aguirre3

  • 1Department of Biomedical Sciences, State University of New York at Albany, Albany, NY, USA.

Molecular and cellular endocrinology
|January 22, 2026
PubMed
概括

针对性腺激素受体的小分子提供了新的避孕和生育治疗选择. 研究揭示了它们在调节受体活性和信号通路以获得精确的治疗效果方面的潜力.

关键词:
其他模拟器的模拟器在GPCRs中,GPCRs是指GPCR.冠状腺热素受体的受体它们是淋巴激素 (Gonadotropins).小分子激动剂小分子激动剂小分子抗剂的作用.

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