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Updated: Feb 13, 2026

Pre-clinical Evaluation of Tyrosine Kinase Inhibitors for Treatment of Acute Leukemia
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以结构为导向的设计和评估基于佐的PIM-1激酶抑制剂具有有前途的抗癌活性

Aanchal Rathi1, Rajesh K Hadiya2, Md Nayab Sulaimani3

  • 1Department of Biotechnology, Faculty of Life Sciences, Jamia Millia Islamia, New Delhi, India.

Journal of biomolecular structure & dynamics
|February 11, 2026
PubMed
概括

新的oxazolone衍生物被设计为用于癌症治疗的PIM-1激酶抑制剂. 化合物O29在前列腺癌细胞中显示出强大的PIM-1抑制和抗癌活性,显示出治疗潜力.

关键词:
癌症治疗治疗 癌症治疗在PIM-1激酶中,PIM-1激酶的作用是:药物开发是药物的发展.激酶抑制剂 激酶抑制剂奥克萨佐龙的衍生品 奥克萨佐龙衍生品

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