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Updated: Feb 14, 2026

Assays for Validating Histone Acetyltransferase Inhibitors
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通过辅酶A类似物抑制氨酸酸转移酶基因组的抑制

Faidra Voukia1, Nurgül Bilgin1, Steffen Bundgaard Andersen1

  • 1Department of Physics, Chemistry and Pharmacy, University of Southern Denmark, Campusvej 55, 5230 Odense, Denmark.

Molecules (Basel, Switzerland)
|February 13, 2026
PubMed
概括

功能化协酶A类型被开发为强大的基因素酸转移酶 (KATs) 的抑制剂. 这些S-功能化辅酶A衍生物显示出创造针对KAT的化学探针的巨大潜力.

关键词:
通过乙化处理.辅酶A 是一种表观遗传学是指表观遗传学.基因组 基因组 基因组lysine 乙转移酶 的作用.

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