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Updated: Feb 14, 2026

Synthesis and Evaluation of a Ruthenium-based Mitochondrial Calcium Uptake Inhibitor
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基于 (E) -α-Fluorovinylphosphonate可逆式甲素C抑制剂的设计,合成和生物活性

Marcin Kaźmierczak1,2, Monika Bilska-Markowska1, Katarzyna Wiśniewska1

  • 1Faculty of Chemistry, Adam Mickiewicz University in Poznań, Uniwersytetu Poznańskiego 8, Poznań 61-614, Poland.

The Journal of organic chemistry
|February 13, 2026
PubMed
概括

研究人员合成了新的基酸二,作为潜在的甲素C抑制剂. 分子对接和活性测试揭示了酶抑制剂设计的有前途的结构特征.

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