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Updated: Feb 25, 2026

Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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Published on: June 13, 2022

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用二次性二乙胺酸进行灾难选择性循环化,以获得endo-Azabicyclo[3.1.0]hexane-6-carboxamides

Terrence-Thang H Nguyen1, Takeru Saito1, Warren Chang1

  • 1Department of Chemistry, Emory University, Atlanta, Georgia 30322, United States.

Organic letters
|February 23, 2026
PubMed
概括

迪罗 (II) 催化剂使烯酸与二乙胺的二选择性循环化成为可能,产生内-azabicyclo[3.1.0]hexane-6-carboxamides. 这种方法对于合成像Mazisotine这样的候选药物至关重要.

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