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Updated: Feb 28, 2026

Reverse Yeast Two-hybrid System to Identify Mammalian Nuclear Receptor Residues that Interact with Ligands and/or Antagonists
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Published on: November 15, 2013

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针对核受体的治疗方法:通过TRβ,ERRα和LXR调节器重编程新陈代谢.

Carmen Di Giovanni1, Antonio Lavecchia1

  • 1"Drug Discovery" Laboratory, Department of Pharmacy, University of Naples Federico II, I-80131 Naples, Italy.

Biomolecules
|February 27, 2026
PubMed
概括

针对TRβ,ERRα和LXR等核受体,为代谢障碍提供了一种新的精确医学方法. 调节剂在治疗脂肪肝疾病,肥胖和脂质失调方面表现有前途,恢复代谢健康.

关键词:
与雌激素相关的受体α.肝脏的X受体是一个X受体.代谢障碍 代谢障碍 代谢障碍线粒体生物发生是线粒体生物发生.非酒精性脂肪性肝病是非酒精性脂肪性肝病.核受体是一种核受体.小分子调节器的小分子调节器.有针对性的治疗.甲状腺激素受体β是甲状腺激素的受体.

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