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Updated: Feb 28, 2026

Facile Preparation of 4-Substituted Quinazoline Derivatives
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通过协同 Pd/Enamine 催化剂实现的抗微生物昆衍生物的合成:实验和计算研究

Mostafa Sayed1, Ahmed Dewan2, Ahmed A El-Rashedy3,4

  • 1Chemistry Department, Faculty of Science, New Valley University, El-Kharja 72511, Egypt.

Precision chemistry
|February 27, 2026
PubMed
概括

研究人员开发了一种新的Pd-(II) /氨基合作催化剂,用于形成C-C键. 五种氨酸衍生物显示出显著的抗微生物活性,得到分子对接和模拟的支持,表明新药开发的潜力.

关键词:
在 Pd 催化剂.氨基胺是一种氨基胺.抗微生物活性的抗微生物活性.昆氨酸 (quinoline) 是一种氨酸.综合合成是一种合成.

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