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Updated: Mar 3, 2026

Optimizing the Genetic Incorporation of Chemical Probes into GPCRs for Photo-crosslinking Mapping and Bioorthogonal Chemistry in Live Mammalian Cells
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量子生物化学 洞察在a1A-腺素受体中的配体识别

Luana Talinne da Costa Gomes1, Katyanna Sales Bezerra2, Elaine Cristina Gavioli1

  • 1Department of Biophysics and Pharmacology, Federal University of Rio Grande Do Norte, Natal 59072-970, Rio Grande do Norte, Brazil.

ACS omega
|March 2, 2026
PubMed
概括

量子生物化学方法准确地预测了连接物与α-1A腺受体 (α1A-AR) 的结合. 这项研究揭示了关键的分子相互作用,有助于设计针对α1A-AR相关疾病的选择性药物.

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