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Updated: Mar 4, 2026

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

Published on: January 21, 2020

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可切换的N-Hvs. 这是一个可切换的N-H. 使用双重功能的试剂进行 C3-H 炭化

Katherine E Marris1, Jazmine T Thorne1, Daniel J Ryder-Mahoney1

  • 1School of Chemistry and Chemical Engineering, University of Southampton, Southampton, SO17 1BJ, UK. gregory.perry@soton.ac.uk.

Chemical communications (Cambridge, England)
|March 3, 2026
PubMed
概括

这项研究引入了一种新的二氧化碳转移反应,用于碳氧化醇和氨基. 反应条件控制N-H或C3-H碳素化是否发生,使重要化合物的合成成为可能.

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