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Updated: May 10, 2026

High-throughput Screening for Small-molecule Modulators of Inward Rectifier Potassium Channels
10:07

High-throughput Screening for Small-molecule Modulators of Inward Rectifier Potassium Channels

Published on: January 27, 2013

大麻二醇通过不同的部位抑制人类的KV7.1和KV7.1/KCNE1通道

A S Kusay1,2, M Pökl3, I Hiniesto-Iñigo3

  • 1Department of Biomedical and Clinical Sciences, Linköping University, SE-581 85, Linköping, Sweden. ali.kusay@liu.se.

Acta pharmacologica Sinica
|March 3, 2026
PubMed
概括

大麻素 (CBD) 结合于KV7.1和KV7.1/KCNE1通道的不同部位,解释了其多样化的作用. 这一发现有助于开发具有较少副作用的选择性KV7调节器.

关键词:
KCNE1 的意思是KCNQ1 一个国家.绑定网站 绑定网站在Cannabidiol中使用.电力生理学 电力生理学分子建模分子建模

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