用酸修饰的PSMA向性-药物合物用于长效前列腺癌治疗

Ziwen Qiu1,2, Xiaorui Zheng2, Shoumei Pan2

  • 1Department of Pulmonary and Critical Care Medicine, Zhujiang Hospital, Southern Medical University Guangzhou 510280 China chen_xin1020@163.com.

Chemical science
|March 12, 2026
PubMed
概括

一种新的酸改性-药物联合体 (PDC) 针对前列腺特异性膜抗原 (PSMA) 来增强前列腺癌治疗. 这种长效的PDC显著改善了药理动力学和瘤抑制,同时减少了副作用.