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Updated: Mar 18, 2026

Pre-clinical Evaluation of Tyrosine Kinase Inhibitors for Treatment of Acute Leukemia
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为抗癌应用设计,合成和生物评估erlotinib-1,2,3-triazole衍生物

Qiyan Yao1, Kexin Qu1, Lan Wang1

  • 1College of Basic Medicine and Forensic Medicine, Henan University of Science and Technology China sanqiangli2001@163.com.

RSC medicinal chemistry
|March 16, 2026
PubMed
概括

新的erlotinib衍生物在肝细胞癌 (HCC) 治疗中显示出有前途. 化合物3d在体外和体内表现出显著的抗瘤活性,毒性最小,这表明它有可能成为HCC的新治疗剂.

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