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Drug-induced Sensitization of Adenylyl Cyclase: Assay Streamlining and Miniaturization for Small Molecule and siRNA Screening Applications
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药理应激光学扫描使用2-环基甲基立基氨酸 (WRC-0470). 一种新型的,短效的腺A2A受体激动剂

D K Glover1, M Ruiz, J Y Yang

  • 1Department of Medicine, University of Virginia Health Sciences Center, Charlottesville 22908, USA. dkg2w@virginia.edu

Circulation
|October 1, 1996
PubMed
概括

一种新的选择性腺A2A受体激动剂,WRC-0470,有效地扩大冠状动脉用于压力成像,而不会引起副作用. 这为接受药理应力测试的患者提供了更安全的替代方案.

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