Related Experiment Videos

Selective inhibition of nuclear steroid receptor function by a protein from a human tumorigenic poxvirus

N Chen1, T Baudino, P N MacDonald

  • 1Department of Molecular Microbiology and Immunology, Saint Louis University Health Sciences Center, St. Louis, Missouri 63104, USA.

Virology
|August 11, 2000
PubMed

Insights

Molluscum contagiosum virus protein MC013L blocks vitamin D and glucocorticoid receptors, potentially aiding viral replication by inhibiting keratinocyte differentiation. This discovery introduces a new class of poxvirus proteins modulating nuclear receptors.

Area of Science:

  • Virology
  • Molecular Biology
  • Dermatology

Background:

  • Molluscum contagiosum (MC) is a widespread viral infection with increasing prevalence.
  • The virus, molluscum contagiosum virus (MCV), utilizes various proteins to manipulate host cell functions for replication.

Purpose of the Study:

  • To investigate the interaction of MCV protein MC013L with host nuclear receptors.
  • To elucidate the role of MC013L in modulating keratinocyte differentiation and its implications for MCV replication.

Main Methods:

  • Yeast two-hybrid assays to detect protein-protein interactions.
  • GST pull-down assays to confirm direct binding.
  • Far Western blot analysis to validate interactions.
  • Analysis of nuclear receptor transactivation inhibition.

Main Results:

  • MCV MC013L protein directly interacts with glucocorticoid receptor (GR) and vitamin D receptor (VDR).
  • MC013L inhibits transactivation mediated by GR and VDR, but not by retinoid or estrogen receptors.
  • Glucocorticoids inhibit keratinocyte proliferation; Vitamin D and retinoids regulate differentiation.

Conclusions:

  • MC013L may promote MCV replication by blocking keratinocyte differentiation through inhibition of GR and VDR signaling.
  • MC013L represents a novel class of poxvirus proteins that directly modulate nuclear receptor-mediated transcription.

Related Concept Videos