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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
07:30

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

Published on: January 21, 2020

A study on the conversion of indanones into carbostyrils

Yasuhiro Torisawa1, Takao Nishi, Jun ichi Minamikawa

  • 1Process Research Laboratory, Second Tokushima Factory, Otsuka Pharmaceutical Co., Ltd., Kawauchi, Tokushima, 771-0182, Japan. torisawa@fact.otsuka.co.jp

Bioorganic & Medicinal Chemistry
|April 26, 2003
PubMed

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