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Updated: Aug 24, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
07:16

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

Selective, orally active gamma-aminobutyric acidA alpha5 receptor inverse agonists as cognition enhancers

Francine Sternfeld1, Robert W Carling, Richard A Jelley

  • 1The Neuroscience Research Centre, Merck Sharp and Dohme Research Laboratories, Terlings Park, Eastwick Road, Harlow, Essex, CM20 2QR, UK. francine_sternfeld@merck.com

Journal of Medicinal Chemistry
|April 16, 2004
PubMed

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