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Updated: Aug 17, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
07:16

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

Efficient synthesis of a GABA A alpha2,3-selective allosteric modulator via a sequential Pd-catalyzed cross-coupling

Mark S Jensen1, R Scott Hoerrner, Wenjie Li

  • 1Department of Process Research, Merck Research Laboratories, P.O. Box 2000, Rahway, NJ 07065, USA. mark_jensen@merck.com

The Journal of Organic Chemistry
|July 16, 2005
PubMed

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