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Updated: Aug 15, 2026

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Transforming bivalent ligands into retractable enzyme inhibitors through polypeptide-protein interactions

Dmitri Tolkatchev1, Anna Vinogradova, Feng Ni

  • 1Bio-NMR and Protein Research Group, Biotechnology Research Institute, National Research Council of Canada, 6100 Royalmount Avenue, Montreal, Que., Canada H4P 2R2.

Bioorganic & Medicinal Chemistry Letters
|October 6, 2005
PubMed

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