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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A potent nonpeptide antagonist of the substance P (NK1) receptor

R M Snider1, J W Constantine, J A Lowe

  • 1Department of Exploratory Medicinal Chemistry, Central Research Division, Pfizer Inc., Groton, CT 06340.

Science (New York, N.Y.)
|January 25, 1991
PubMed

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