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Updated: Jul 13, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Allosteric GPCR modulators: taking advantage of permissive receptor pharmacology

Katie Leach1, Patrick M Sexton, Arthur Christopoulos

  • 1Drug Discovery Biology Laboratory, Department of Pharmacology, Monash University, Clayton, Victoria 3800, Australia.

Trends in Pharmacological Sciences
|July 17, 2007
PubMed

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