Identification and optimization of a novel series of [2.2.1]-oxabicyclo imide-based androgen receptor antagonists

Mark E Salvati1, Aaron Balog, Weifang Shan

  • 1Department of Oncology Chemistry, Bristol-Myers Squibb Pharmaceutical Research and Development, PO Box 4000, Princeton, NJ 08543-4000, USA. mark.salvati@bms.co

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