Related Experiment Video

Updated: Jul 6, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

Allosteric modulation of kinases and GPCRs: design principles and structural diversity

Jana A Lewis1, Evan P Lebois, Craig W Lindsley

  • 1Department of Pharmacology and Chemistry, Vanderbilt Program in Drug Discovery, Vanderbilt Institute of Chemical Biology, Vanderbilt University Medical Center, Nashville, TN 37232-6600, USA. jana.a.lewis@vanderbilt.edu

Current Opinion in Chemical Biology
|March 18, 2008
PubMed

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