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Preparation of N-(2-alkoxyvinyl)sulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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A simple, modular method for the synthesis of 3,4,5-trisubstituted pyrazoles

Mark McLaughlin1, Karen Marcantonio, Cheng-Yi Chen

  • 1Process Research, Merck Research Laboratories, Rahway, NJ 07065, USA. mark_mclaughlin@merck.com

The Journal of Organic Chemistry
|May 1, 2008
PubMed

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