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Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines
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Discovery of brain penetrant, soluble, pyrazole amide EP1 receptor antagonists

Adrian Hall1, Andy Billinton, Alan K Bristow

  • 1Neurolosciences Centre of Excellence for Drug Discovery, GlaxoSmithKline, New Frontiers Science Park, Third Avenue, Harlow, Essex CM19 5AW, UK. adrian.2.hall@gsk.com

Bioorganic & Medicinal Chemistry Letters
|June 24, 2008
PubMed

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