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Taranabant, a novel cannabinoid type 1 receptor inverse agonist

Bradley A Fremming1, Steven T Boyd

  • 1University of Nebraska Medical Center, College of Medicine, Michael F Sorrell Center for Health Science Education, 15926 S St, Omaha, NE 68135, USA. bfremming@unmc.edu

Current Opinion in Investigational Drugs (London, England : 2000)
|September 30, 2008
PubMed
Summary

Merck & Co Inc is developing taranabant, a cannabinoid receptor type 1 inverse agonist, for obesity and nicotine dependence. Clinical trials are underway, with Phase III for obesity and completed Phase II for smoking cessation.

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