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Assays for Validating Histone Acetyltransferase Inhibitors
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SAR profiles of spirocyclic nicotinamide derived selective HDAC1/HDAC2 inhibitors (SHI-1:2)

Joey L Methot1, Christopher L Hamblett, Dawn M Mampreian

  • 1Department of Drug Design and Optimization, Merck Research Laboratories, 33 Avenue Louis Pasteur, Boston, MA 02115, USA. joey_methot@merck.com

Bioorganic & Medicinal Chemistry Letters
|October 28, 2008
PubMed

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