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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

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Synthesis and preliminary screening of novel indole-3-methanamines as 5-HT4 receptor ligands

Amir Hanna-Elias1, David T Manallack, Isabelle Berque-Bestel

  • 1Medicinal Chemistry and Drug Action, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.

European Journal of Medicinal Chemistry
|February 19, 2009
PubMed

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