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A Method for Screening and Validation of Resistant Mutations Against Kinase Inhibitors
12:40

A Method for Screening and Validation of Resistant Mutations Against Kinase Inhibitors

Published on: December 7, 2014

2-Aminopyrazolo[1,5-a]pyrimidines as potent and selective inhibitors of JAK2

Mark W Ledeboer1, Albert C Pierce, John P Duffy

  • 1Vertex Pharmaceuticals Inc, Cambridge, MA 02139-4242, United States. mark_ledeboer@vrtx.com

Bioorganic & Medicinal Chemistry Letters
|October 28, 2009
PubMed

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