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4-methylpteridinones as orally active and selective PI3K/mTOR dual inhibitors

Kevin K-C Liu1, Shubha Bagrodia, Simon Bailey

  • 1Pfizer Global Research and Development, Chemistry Department, La Jolla, CA 92120, USA. kevin.k.liu@pfizer.com

Bioorganic & Medicinal Chemistry Letters
|September 7, 2010
PubMed

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