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Preparation of N-(2-alkoxyvinyl)sulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Trifluoromethylphenyl as P2 for ketoamide-based cathepsin S inhibitors

Jiaqiang Cai1, John Robinson, Simone Belshaw

  • 1Merck Research Laboratories, MSD, Newhouse, Lanarkshire, United Kingdom. jiaqiang.cai@merck.com

Bioorganic & Medicinal Chemistry Letters
|October 30, 2010
PubMed

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