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From KRASG12D to Pan-KRAS Inhibitors─A Journey Enabled by Synthetic Innovation and Structure-Based Drug Design

Xiaoshen Ma1, David L Sloman1, Timothy J Henderson1

  • 1Department of Discovery Chemistry, Merck & Co., Inc., 33 Ave. Louis Pasteur, Boston 02215, Massachusetts, United States.

Journal of Medicinal Chemistry
|April 9, 2026
PubMed

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