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Updated: May 23, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Discovery of a potent and selective GPR120 agonist

Bharat Shimpukade1, Brian D Hudson, Christine Kiel Hovgaard

  • 1Department of Physics, Chemistry and Pharmacy, University of Southern Denmark, Campusvej 55, DK-5230 Odense M, Denmark.

Journal of Medicinal Chemistry
|April 24, 2012
PubMed

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