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Reverse Yeast Two-hybrid System to Identify Mammalian Nuclear Receptor Residues that Interact with Ligands and/or Antagonists
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Discovery and optimization of a series of liver X receptor antagonists

XianYun Jiao1, David J Kopecky, Ben Fisher

  • 1Department of Medicinal Chemistry, Amgen Inc., 1120 Veterans Blvd., South San Francisco, CA 94080, USA. xjiao@amgen.com

Bioorganic & Medicinal Chemistry Letters
|August 21, 2012
PubMed

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