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Chemical Inactivation of the E3 Ubiquitin Ligase Cereblon by Pomalidomide-based Homo-PROTACs
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Chemical Inactivation of the E3 Ubiquitin Ligase Cereblon by Pomalidomide-based Homo-PROTACs

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UNC1062, a new and potent Mer inhibitor

Jing Liu1, Weihe Zhang, Michael A Stashko

  • 1Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, NC 27599, USA.

European Journal of Medicinal Chemistry
|May 23, 2013
PubMed
Abstract

Keywords:
GlioblastomaKAAPXWSYROPAEL-GUAVBDGJSA-NLeukemiaMer inhibitorsNon-small cell lung cancerPyrazolopyrimidinesSulfonamides

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