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Updated: May 6, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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G protein-coupled receptor transactivation: from molecules to mice

Kim C Jonas1, Adolfo Rivero-Müller, Ilpo T Huhtaniemi

  • 1Department of Surgery and Cancer, Institute of Reproductive and Developmental Biology, Imperial College London, London, United Kingdom.

Methods in Cell Biology
|October 23, 2013
PubMed

Keywords:
BACDimerGPCRGonadotropinLuteinizing hormoneMouse modelReproductionSignalingTransactivation

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