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Updated: May 3, 2026

Reverse Yeast Two-hybrid System to Identify Mammalian Nuclear Receptor Residues that Interact with Ligands and/or Antagonists
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Binding mode and structure-activity relationships around direct inhibitors of the Nrf2-Keap1 complex

Eric Jnoff1, Claudia Albrecht, John J Barker

  • 1UCB Pharma, UCB NewMedicines, Chemin du Foriest, 1420 Braine-l'Alleud (Belgium). eric.jnoff@ucb.com.

Chemmedchem
|February 8, 2014
PubMed

Keywords:
CNSKeap1Nrf2co-crystal structuresdockingstructure-activity relationships

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