A fragment-based approach to identifying S-adenosyl-l-methionine -competitive inhibitors of catechol O-methyl

Marion Lanier1, Geza Ambrus, Derek C Cole

  • 1Medicinal Chemistry, ‡Structural Biology, §Discovery Biology, ∥Analytical Chemistry, Takeda California Inc. , 10410 Science Center Drive San Diego California 92121, United States.