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Updated: Apr 28, 2026

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Design of a Potent CB1 Receptor Antagonist Series: Potential Scaffold for Peripherally-Targeted Agents

Robert L Dow1, Philip A Carpino1, Denise Gautreau1

  • 1Pfizer Worldwide Research and Development , Eastern Point Road, Groton, Connecticut 06340, United States.

ACS Medicinal Chemistry Letters
|June 6, 2014
PubMed

Keywords:
Obesityantagonistcannabinoid receptorclearanceligand efficiencyligand-lipophilicity efficiencymultidrug resistance protein 1polar surface area

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