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Updated: Apr 28, 2026

Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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Chiral Resolution and Serendipitous Fluorination Reaction for the Selective Dopamine D3 Receptor Antagonist BAK2-66

Vivek Kumar1, Ashwini K Banala1, Erick G Garcia1

  • 1Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse-Intramural Research Program, National Institutes of Health , 333 Cassell Drive, Baltimore, Maryland 21224, United States.

ACS Medicinal Chemistry Letters
|June 20, 2014
PubMed

Keywords:
DASTasymmetric catalysisdopamineenantioselectivity

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