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Thermostabilization, Expression, Purification, and Crystallization of the Human Serotonin Transporter Bound to S-citalopram
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Thermostabilization, Expression, Purification, and Crystallization of the Human Serotonin Transporter Bound to S-citalopram

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Novel and high affinity fluorescent ligands for the serotonin transporter based on (s)-citalopram

Vivek Kumar1, Troels Rahbek-Clemmensen2, Christian B Billesbølle2

  • 1Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse-Intramural Research Program, National Institutes of Health , 333 Cassell Drive, Baltimore, Maryland 21224, United States.

ACS Medicinal Chemistry Letters
|June 20, 2014
PubMed

Keywords:
Fluorescent ligandSERTcitalopramrhodamine

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