Benzocoumarins: isolation, synthesis, and biological activities

Hai-Ning Lv, Peng-Fei Tu, Yong Jiang1

  • 1State Key Laboratory of Natural and Biomimetic Drugs, Peking University, Beijing 100191, China. yongjiang@bjmu.edu.cn.

Summary

This review summarizes benzocoumarin research from 1953-2014, covering isolation, synthesis, and biological activities of these coumarin derivatives. Efforts focus on novel analogs with enhanced bioactivities and improved synthetic methods.

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