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A High-throughput Calcium-flux Assay to Study NMDA-receptors with Sensitivity to Glycine/D-serine and Glutamate
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Tryptophanol-derived oxazolopiperidone lactams: identification of a hit compound as NMDA receptor antagonist

Nuno A L Pereira1, Francesc X Sureda2, Roser Esplugas2

  • 1Instituto de Investigação do Medicamento (iMed.ULisboa), Faculdade de Farmácia, Universidade de Lisboa, Av. Prof. Gama Pinto, 1649-003 Lisboa, Portugal.

Bioorganic & Medicinal Chemistry Letters
|June 30, 2014
PubMed

Keywords:
N-Methyl-d-aspartate receptorsNMDAR antagonistNeurodegenerative diseasesOxazolopiperidonesTryptophanol

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