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Discovery of Spiro[cyclohexane-dihydropyrano[3,4-b]indole]-amines as Potent NOP and Opioid Receptor Agonists

Stefan Schunk1, Klaus Linz1, Sven Frormann1

  • 1Departments of Medicinal Chemistry, Preclinical Drug Safety, Molecular Pharmacology, Pain Pharmacology, Pharmacokinetics, and Discovery Informatics, Global Drug Discovery, Grünenthal Innovation, Grünenthal GmbH , D-52099 Aachen, Germany.

ACS Medicinal Chemistry Letters
|August 23, 2014
PubMed

Keywords:
MOP receptor agonistNOP receptor agonist

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